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Publications

Bertin, M. J.; Demirkiran, O.; Navarro, G.; Moss, N. A.; Lee, J.; Goldgof, G. M.; Vigil, E.; Winzeler, E. A.; Valeriote, F. A.; Gerwick, W. H. “Kalkipyrone B, a marine cyanobacterial γ-​pyrone possessing cytotoxic and anti-​fungal activities.” Phytochemistry 2016, 122, 113-118.

Lassalas, P.; Gay, B.; Lasfargeas, C.; James, M. J.; Tran, V.; Vijayendran, K. G.; Brudent, K. R.; Kozlowski, M. C.; Thomas, C. J.; Smith, A. B. III; Huryn, D. M.; Ballatore, C. “Structure property relationships of carboxylic isosteres.” J. Med. Chem. 2016, 59, 3183-3203.

Johnson, T. C.; Chin, M. R.: Han, T.; Shen, J. P.; Rana, T.; Siegel, D. “Synthesis of Eupalinilide E a Promoter of Human Hematopoietic Stem and Progenitor Cell Expansion.” J. Am. Chem. Soc. 2016, 138, 6068-6073.

Sapkota, M.; Li, Liang; Choi, H.; Gerwick, W. H.; Soh, Y. Bromo-​honaucin A inhibits osteoclastogenic differentiation in RAW 264.7 cells via Akt and ERK signaling pathways.” European Journal of Pharmacology 2015, 769, 100-109.

Miller, B.; Friedman, A. J.; Choi, H.; Hogan, J.; McCammon, J. A.; Hook, V.; Gerwick, W. H. “The marine cyanobacterial metabolite gallinamide A is a potent and selective inhibitor of human cathepsin L.” J. Nat. Prod. 2014, 77, 92-99.

Lou, K.; Yao, Y.; Hoye, A. T. James, M. J.; Cornec, A. S.; Hyde, E.; Gay, B.; Lee, V. M.; Trojanowski, J. Q.; Smith, A. B. III; Bruden, K. R.; Ballatore, C. “Brain-penetrant, orally bioavailable microtubule-stabilizing small molecules are potential candidate therapeutics for Alzheimer's disease and related tauopathies.” J. Med. Chem. 2014, 57, 6116-6127.

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